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PHARMA INTERMEDIATES

API  Intermediate Name CAS No.
ApixabanAcetic acid, 2-chloro-2-[2-(4-methoxyphenyl)hydrazinylidene], ethyl ester27143-07-3
Apixaban3-Morpholino-1-(4-nitrophenyl)-5,6-dihydropyridin-2(1H)-one545445-44-1
ABT-888
(S)-2-Methylproline42856-71-3
Acalabrutinib(3-Chloropyrazin-2-yl)MethanaMine hydrochloride939412-86-9
AcalabrutinibN-Benzyloxycarbonyl-L-proline1148-11-4
AcalabrutinibN-Pyridin-2-yl-4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-benzamide1383385-64-5
Acalabrutinib2-Butynoic acid590-93-2
Abiraterone Acetate17-Iodoandrosta-5,16-dien-3beta-ol32138-69-5
Abiraterone Acetate17-Iodoandrosta-5,16-dien-3beta-ol 3-acetate114611-53-9
Canagliflozin
2-(4-FLUOROPHENYL)THIOPHENE58861-48-6
Canagliflozin5-Bromo-2-methylbenzoic acid79669-49-1
Canagliflozin2-(4-Fluorophenyl)-5-[(5-iodo-2-methylphenyl)methyl]thiophene898566-17-1
Ceritinib/Crizotinib4-(4-Bromopyrazol-1-yl)piperidine-1-carboxylic acid tert-butyl ester877399-50-3
Ceritinib/Crizotinibtert-Butyl 4-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]piperidine-1-carboxylate877399-74-1
Ceritinib/Crizotinib(S)-1-(2,6-Dichloro-3-fluorophenyl)ethanol877397-65-4;42247-74-5
Ceritinib/Crizotinib(R)-5-bromo-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)pyridin-2-amine877399-00-3
ClopidogrelThiophene-2-ethanol5402-55-1
Clopidogrel4,5,6,7-Tetrahydro-thieno[3,2-c]pyridine HCl28783-41-7
Docetaxel10-Deacetylbaccatin III32981-86-5
Duloxetine(S)-(-)-N,N-Dimethyl-3-hydroxy-3-(2-thienyl)propanamine132335-44-5
Entecavir6-(Benzyloxy)-9-((1S,3R,3S)-4-(benzyloxy)-3-(benzyloxymethyl)-2-methylenecyclopentyl)-N-((4-methoxyphenyl)diphenylmethyl)-9H-purin-2-amine142217-80-9
Ezetimibe(3R,4S)-4-(4-(Benzyloxy)Phenyl)-1-(4-Fluorophenyl)-3-((S)-3-(4- Fluorophenyl)-3-Hydroxypropyl)Azetidin-2-One163222-32-0
EdoxabanEthyl 2-((5-chloropyridin-2-yl)amino)-2-oxoacetate hydrochloride1243308-37-3
Edoxaban5-Methyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine-2-carboxylic acid hydrochloride720720-96-7
EdoxabanTert-Butyl(1R,2S,5S)-2-azido-5-[(dimethylamino)carbonyl]cyclohexylcarbamate oxalic acid1353893-22-7
Elagolix1-[2-fluoro-6-(trifluoromethyl)benzyl]-5-iodo-6-methylpyrimidine-2,4(1H,3H)-dione1150560-54-5
Elagolix(R)-N-(tert-Butoxycarbonyl)-2-phenylglycinol102089-74-7
Elagolix2-FLUORO-3-METHOXYPHENYLBORONIC ACID352303-67-4
Empagliflozin(3S)-3-[4-[(5-Bromo-2-chlorophenyl)methyl]phenoxy]tetrahydro-furan915095-89-5
Famciclovir9-(4-Acetoxy-3-acetoxymethylbutyl)-2-amino-6-chloropurine97845-60-8
Linagliptin8-bromo-7-(but-2-ynyl)-3-methyl-1H-purine-2,6(3H,7H)-dione666816-98-4
Linagliptin2-(chloromethyl)-4-methylquinazoline109113-72-6
Linagliptin8-Bromo-7-but-2-ynyl-3-methyl-1-(4-methyl-quinazolin-2-ylmethyl)-3,7-dihydro-purine-2,6-dione853029-57-9
Lenvatinib4-chloro-7-methoxyquinoline-6-carboxamide417721-36-9
Lenvatinib4-Amino-3-chlorophenol hydrochloride52671-64-4
LevetiracetamL-2-aminobutanamide HCl7682-20-4
Lusutrombopag(E)-3,5-dichloro-4-(3-ethoxy-2-methyl-3-oxoprop-1-enyl)benzoic acid1110767-89-9
Lusutrombopag(S)-4-(3-(1-(hexyloxy)ethyl)-2-methoxyphenyl)thiazol-2-amine1110767-98-0
Meropenem
4AA: 4-Acetoxy-2-azetidinone28562-53-0
MeropenemMAP (Beta-Methyl vinyl phosphate)90776-59-3
Neratinib
3-chloro-4-(pyridin-2-ylmethoxy)aniline524955-09-7
NeratinibN-(4-Chloro-3-cyano-7-ethoxy-6-quinolinyl)acetamide848133-76-6
Neratinib6-amino-4-(3-chloro-4-(pyridin-2-ylmethoxy)phenylamino)-7-ethoxyquinoline-3-carbonitrile848139-78-6
Neratinibtrans-4-Dimethylaminocrotonic acid hydrochloride848133-35-7
Nilotinib
3-(4-Methyl-1H-imidazol-1-yl)-5-(trifluoromethyl)aniline641571-11-1
NilotinibDiphenylphosphoryl azide26386-88-9
Nilotinib4-Methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]benzoic acid641569-94-0
Nilotinib1-(3-Pyridyl)-3-(dimethylamino)-2-propen-1-one55314-16-4
Olmesartan
5-(4'-Bromomethyl-1,1'-biphenyl-2-yl)-1-triphenylmethyl-1H-tetrazole124750-51-2
OlmesartanEthyl 4-(1-hydroxy-1-methylethyl)-2-propyl-imidazole-5-carboxylate144689-93-0
Olmesartan1-(4-ethoxycarbonylphenyl)pyrrole144690-33-5
Palbociclibtert-butyl 4-(6-amino-3-pyridyl)piperazine-1-carboxylate571188-59-5
Palbociclib6-Bromo-2-chloro-8-cyclopentyl-5-methylpyrido[2,3-d]pyrimidin-7(8H)-one1016636-76-2
Pregabalin3-Carbamoymethyl-5-methylhexanoic acid181289-15-6
Ribociclib2-Chloro-7-cyclopentyl-n,n-dimethyl-7h-pyrrolo[2,3d]pyrimidine-6-carboxamide1211443-61-6
Ribociclib2-Chloro-7-cyclopentyl-7H-pyrrolo[2,3-d]pyrimidine-6-carboxylic acid1211443-58-1
Rivaroxaban4-(4-Aminophenyl)morpholin-3-one438056-69-0
Rivaroxaban5-Chlorothiophene-2-carboxylic acid24065-33-6
Rivaroxaban
(S)-(+)-N-(2,3-Epoxypropyl)phthalimide161596-47-0
RosuvastatinZ-9: 4-(4-Fluorophenyl)-6-Isopropyl-2-[(N-methyl-N-methylsulfonyl)amino] pyrimidinyl-5-yl-formyl147118-37-4
RosuvastatinZ-7: 4-(4-Fluorophenyl)-6-isopropyl-2-[(N-methyl-N-methylsufonyl)amino]pyrimidine-5-yl-methanol147118-36-3
Sotagliflozin4-Iodo-1-chloro-2-(4-ethoxybenzyl)benzene1103738-29-9
SotagliflozinD-xylo-Pentodialdo-5,2-furanose, 4,5-O-(1-Methylethylidene)-1-C-4-Morpholinyl-,(5S)-1103738-19-7
SotagliflozinD-xylo-Pentodialdo-5,2-furanose, 1-C-[4-chloro-3-[(4-ethoxyphenyl)Methyl]phenyl]-4,5-O-(1-Methylethylidene)-,(5S)-1103738-30-2
Sotagliflozin5-bromo-2-chloro-4’-ethoxydiphenylmethane461432-23-5
Saxagliptin(1S,3S,5S)-3-(Aminocarbonyl)-2-azabicyclo[3.1.0]hexane-2-carboxylic acid tert-butyl ester361440-67-7
Saxagliptin(alphaS)-alpha-[[(1,1-Dimethylethoxy)carbonyl]amino]-3-hydroxytricyclo[3.3.1.13,7]decane-1-acetic acid361442-00-4
SaxagliptinLCZ6961426129-50-1
Saxagliptin(2R,4S)-5-([1,1'-biphenyl]-4-yl)-4-((tert-butoxycarbonyl)aMino)-2-Methylpentanoic acid1012341-50-2
AHU377149709-62-6
Sacubitril2,4,5-Trifluorophenylacetic acid209995-38-0
SacubitrilBoc-(R)-3-Amino-4-(2,4,5-Trifluoro-Phenyl)-Butyric Acid486460-00-8
Sacubitril3-(Trifluoromethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazine hydrochloride762240-92-6
Tofacitinib4-Chloro-7H-pyrrolo[2,3-d]pyrimidine3680-69-1
Tofacitinib(3R,4R)-N,4-Dimethyl-1-(phenylmethyl)-3-piperidinamine hydrochloride1062580-52-2
Telaprevir(2S)-2-Cyclohexyl-N-(2-pyrazinylcarbonyl) glycyl-3-methyl-L-valine402958-96-7
Ticagrelor2-((3aR,4S,6R,6aS)-6-amino-2,2-dimethyltetrahydro-3aH-cyclopenta[d][1,3]dioxol-4-yloxy)ethanol L-tataric acid376608-65-0
Ticagrelor(1R,2S)-2-(3,4-Difluorophenyl)cyclopropanaminium(2R)-hydroxy(phenyl)ethanoate376608-71-8
TicagrelorCyclopropanamine,2-(3,4-difluorophenyl)-(1R,2S) -(2R,3R)-2,3-dihydroxybutanedioate220352-39-6
Ticagrelor4,6-dichloro-2-propylthiopyrimidine-5-amine145783-15-9
Upadacitinib5-Bromo-4,7-diazaindole875781-43-4
VildagliptinL-Prolinamide7531-52-4
Vildagliptin(2S)-1-(Chloroacetyl)-2-pyrrolidinecarbonitrile207557-35-5
Alfuzosin / Terazosin(N-[3-[(4-Amino-6,7-dimethoxy-2-quinazolynyl)methylaminopropyl]tetrahydro-2-furancarboxamide] ▲81403-80-7
Alfuzosin / Terazosin4-Amino-2-chloro-6,7-dimethoxyquinazoline ▲23680-84-4
PatiromerMethyl 2-Fluoroacrylate ▲2343-89-7
Quinapril(S)-1,2,3,4-Tetrahydro-3-isoquinolinecarboxylic acid ▲74163-81-8
FenofibrateFenofibrate acid: (2-[4-(4-chlorobenzoyl)phenoxy]-2-methylpropionic acid) ▲42017-89-0
Empagliflozin2,3,4,6-Tetrakis-O-trimethylsilyl-D-gluconolactone ▲32384-65-9
Triamterene5-NITROSO-2,4,6-TRIAMINOPYRIMIDINE ▲1006-23-1
Tofacitinib4-CHLORO-7H-PYRROLO (2,3-D) PYRIMIDINE ▲3680-69-1
Tofacitinib4-CHLORO- 7-Tosyl- 7H-PYRROLO[2,3,D]PYRIMIDINE ▲479633-63-1
LacosamideAll intermediates ▲175481-36-4
VildagliptinL-Prolinamide ▲7531-52-4

Others

3-Methyl-4-isopropylphenol ▲3228-02-2
OthersThymol ▲89-83-8
OthersAcetaldehyde oxime ▲107-29-9
OthersHydroxylamine hydrochloride ▲1304222
OthersHydroxylamine sulfate ▲10039-54-0
OthersFAVIPIRAVIR259793-96-9
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